Compile Data Set for Download or QSAR
maximum 50k data
Found 36 of ec50 data for polymerid = 50004809
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50080867(CHEMBL3421671)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli BL21 DE3 after 4 to 6 hrs by GFP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  7nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  7nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351510(CHEMBL8463)
Affinity DataEC50:  10nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351515(CHEMBL1823932)
Affinity DataEC50:  10nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351510(CHEMBL8463)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351513(CHEMBL8450)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468430(CHEMBL4283085)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50080869(CHEMBL1236450)
Affinity DataEC50:  28nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468428(CHEBI:44612 | CHEMBL1234965)
Affinity DataEC50:  30nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  31nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351252(CHEMBL8755)
Affinity DataEC50:  33nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351252(CHEMBL8755)
Affinity DataEC50:  40nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351514(CHEMBL8609)
Affinity DataEC50:  54nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50527017(CHEMBL4461584)
Affinity DataEC50:  71nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468425(CHEBI:56080 | CHEMBL208383)
Affinity DataEC50:  110nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50080868(CHEMBL3421670)
Affinity DataEC50:  119nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli BL21 DE3 after 4 to 6 hrs by GFP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  139nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351511(CHEMBL463321)
Affinity DataEC50:  150nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468427(CHEMBL1812101)
Affinity DataEC50:  162nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468432(CHEMBL4285396)
Affinity DataEC50:  256nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50248862(CHEMBL473592 | N-(3-oxo-3-phenylpropanoyl)-L-homos...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468429(CHEMBL4279608)
Affinity DataEC50:  906nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468424(CHEMBL4287516)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50526977(CHEMBL4462112)
Affinity DataEC50:  2.60E+3nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50527004(CHEMBL4450449)
Affinity DataEC50:  4.20E+3nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350705(CHEMBL1814827)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50527002(CHEMBL4444462)
Affinity DataEC50:  1.70E+4nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350706(CHEMBL1811922)
Affinity DataEC50:  2.10E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50266165((S)-N-(2-oxotetrahydrofuran-3-yl)-2-(4-(trifluorom...)
Affinity DataEC50:  1.40E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351511(CHEMBL463321)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241433((S)-3-(4-bromophenyl)-N-(2-oxo-tetrahydrofuran-3-y...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50527003(CHEMBL4522587)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed